Why does Tapentadol make you sleepy? Know the reason

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Why does Tapentadol make you sleepy? Know the
reason Tapentadol is a medicine used for
treating severe pain. It will only be given if
your doctor considers that other non-opioid
painkillers are ineffective or that you are not
able to tolerate them. Tapentadol is not commonly
prescribed for the management of chronic
(long-term) pain. People who are using tapentadol
are experiencing sleepiness as a side effect. In
this article, we will explore the reasons why
Tapentadol users are experiencing drowsiness and
give insights into its pharmacological effects
Overview and mechanism of action of
tapentadol Tapentadol is a synthetic painkiller
that acts centrally and has a dual mechanism of
action. It is an agonist of the mu-opioid
receptor which additionally inhibits
norepinephrine reuptake. Tapentadol stands apart
from traditional opioids by inhibiting the
reuptake of norepinephrine. Norepinephrine is a
neurotransmitter involved in the body's stress
response and the regulation of wakefulness and
alertness. Tapentadol was approved by the FDA for
the first time in 2008. Later in 2011, the FDA
also approved extended-release tablets of
tapentadol. Tapentadol is used to treat acute
pain that is sufficiently severe for the use of
an opioid painkiller and for which other
therapies are ineffective. Tapentadol is intended
for individuals who have no other treatment
alternatives due to potential risks of addiction,
drug abuse, and drug misuse. Tapentadol
extended-release tablets are intended for the
treatment of pain severe enough to necessitate
daily, around-the-clock pain relievers and for
which alternate treatment options are
unsatisfactory. They are also suggested for the
treatment of neuropathic pain associated with
diabetic peripheral neuropathy (DPN) in people
who require daily, around-the-clock, long-term
opioid medication and for whom alternate
treatment alternatives are insufficient.
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Reasons behind tapentadol to cause
Sleepiness Due to some specific reasons,
tapentadol users feel sleepiness and the reasons
are as follows. The effect of sleepiness The
dual mechanism of action of tapentadol,
especially the inhibition of norepinephrine
reuptake causes sleepiness in tapentadol users.
Because Tapentadol increases the availability of
norepinephrine in the synaptic cleft by blocking
norepinephrine reuptake. The increased levels of
norepinephrine which are known for alertness, can
paradoxically cause drowsiness in some
people. Individual Differences It is essential
to understand that not everyone who takes
Tapentadol will experience the same level of
drowsiness. Individual differences will influence
how the body responds to drugs. The severity of
side effects can be influenced by some other
factors such as overall health, drug tolerance,
and the drug dose. Tapentadol Dose The dose of
tapentadol suggested by your physician is an
important factor in managing adverse effects like
sleepiness. To get the best pain relief while
minimizing side effects, healthcare experts
frequently start treatment with a lower dose and
gradually increase it. Adjusting the dosage may
help in achieving a balance between pain relief
and the side effects including sleepiness.
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Other Things to Think About Tapentadol, like
any medicine, may have other side effects in
addition to drowsiness. Nausea, constipation,
dizziness, and headache are some of the most
commonly seen adverse effects. To manage these
side effects, doctors should adjust the treatment
plan to according individual needs and
conditions. Potential Adverse Effects of
Tapentadol other than Sleepiness Tapentadol,
while useful in pain management, can cause the
following adverse effects Vomiting and
nausea Some people may experience nausea or
vomiting, especially when taking Tapentadol for
the first time. These symptoms can be addressed
by taking the medicine with food or as instructed
by your doctor. Constipation Constipation is a
typical adverse effect of several opioid
medicines. Having enough hydration, including
dietary fiber, and engaging in regular physical
activity will all help to manage this
condition. Lightheadedness and
dizziness Tapentadol might make you dizzy and
lightheaded, especially when you change
positions. Precautions such as gently moving from
a seat or sleeping position may assist in
reducing these consequences. Addiction There
is a chance for dependency because Tapentadol is
an opioid. So it is essential to adhere to
prescribed doses and talk freely with your
healthcare practitioner about any concerns or
changes in your reactions to the medicine. To
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